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Table 1 IC50 Values of eIF4F complex inhibitors

From: The impact of androgen-induced translation in modulating androgen receptor activity

 

Briciclib [nM]

Rocaglamid [nM]

SBI–0640756 [nM]

LNCaP

5.6

32

295

C4-2

2.8

6.7

847

22Rv1

3.3

35

542

Range

1–10

10–100

100–1000